CABASER 2MG – mens health drug, this drug contains Cabergoline and is made by Pharmacia.
Cabergoline is a drug most often medically prescribed for its ability to inhibit prolactin secretion via its action as a dopamine agonist. The drug has been adopted by bodybuilders and strength athletes as a means to combat prolactin related side effects caused by certain anabolic steroids. For this purpose cabergoline is extremely effective while presenting little risk in terms of serious side effects to the health of the user when used for this purpose.
CABASER 2MG is usually employed by bodybuilders to combat prolactin and effects related to prolactin, that’s so before we go any further, lets , it’s very important to understand exactly what that hormone is. Prolactin is a single-chain protein, very closely related to growth hormone. It is secreted by what’s known as lactotrophs in the anterior part of your pituitary gland. In addition, Prolactin is also synthesized and secreted by many other cells in the body, like immune cells, in the brain, and in women is even secreted by the decidua, in the uterus of pregnant women.
If you’ve done any reading at all on prolactin, you have probably come across the fact that its major effects are felt by the mammary gland, and that stimulating mammary gland development and milk production are its primary role. While this is true, many issues have prolactin receptors, and although the anterior pituitary is the major source of prolactin, it is actually synthesized and secreted in several other tissues. Too much prolactin expression can even be responsible for certain types of pituitary tumors. But the most prevalent side effect we see from it in bodybuilders is development of excess mammary tissue and milk production. Unfortunately, mammary gland development and milk production are among its major effects. Great if you are a cow, but not so great if you are a bodybuilder. Yeah, that’s right- too much prolactin can cause galactorrhea. The other prevalent side effect is sexual dysfunction. I suspect that the average male bodybuilder doesn’t want anything to do with any of that.
CABASER 2MG works to inhibit secretion of prolactin because it is a dopamine receptor agonist. This means that it acts upon dopamine receptors in the same way as dopamine does in the body. Dopamine acts as a prolactin inhibitor by binding to receptors in the lactotrophs in the pituitary gland and signals for these to cease the synthesis and secretion of prolactin.
While dopamine exhibits an ability to inhibit the secretion of prolactin it of course has numerous other functions in the body, with CABASER 2MG being able to mimic the action of dopamine and also performing many of these. These functions include creating a sense of wellbeing or contentment via a chemical reaction in the body, most often released during pleasurable or satisfying physical actions. It has even been shown that dopamine-receptor agonists such as Cabergoline can help increase the likelihood that individuals that are quitting smoking be successful. Dopamine can also help improve brain function. For this reason CABASER 2MG is sometimes prescribed to sufferers of Parkinson’s disease. For the average user however it may help in improving memory or even motor functions, although if normal dopamine levels are already being produced by the user this effect will likely be minimal at best. However the primary reason for use of CABASER 2MG by steroid users remains for the treatment of prolactin related side effects.
The anabolic steroids that can lead to excessive levels of prolactin are primarily nandrolone and nandrolone-derived compounds. Steroids such as Deca Durabolin, Trenbolone, and Durabolin all can have this effect. For this reason users of these drugs may want to have a compound such as CABASER 2MG in their possession to treat negative side effects related to prolactin if they should develop at any point during a steroid cycle.
A secondary factor in controlling the levels of prolactin in users of anabolic steroids is the amount of circulating estrogen in their systems. Estrogen has an apparent positive effect on the amount of prolactin produced, with the more estrogen that is produced being related to the amount of prolactin that is produced accordingly. Essentially estrogen stimulates the secretion of prolactin via the disruption of the inhibitory effect of dopamine. For this reason often times prolactin can be controlled by way of the reduction of estrogen levels. Use of aromatase inhibitors can be used for this purpose. However when prolactin levels reach a point where a reduction of estrogen levels does not inhibit excessive prolactin secretion enough, administration of cabergoline should be sufficient to inhibit any further overproduction.
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